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CAS No.: 387867-13-2
Synonyms: MLN518;CT53518;NSC-726292
Tandutinib is an antagonist of FLT3 with IC50 of 0.22 μM and can also inhibit PDGFR and c-Kit thereby inhibiting cellular proliferation and inducing apoptosis.
生物活性
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
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NCT00064584 | Acute Myelogenous Leukemia ... more >> Myelodysplastic Syndrome Collapse << | Phase 1 | Completed | - | United States, California ... more >> UCLA Medical Center Los Angeles, California, United States, 90095 United States, Massachusetts Dana Farber Cancer Institute Boston, Massachusetts, United States, 02115 United States, New York Memorial Sloan Kettering Cancer Center New York, New York, United States, 10021 United States, Ohio Ohio State University Medical Center Columbus, Ohio, United States, 43210 United States, Oregon Oregon Health Sciences University Portland, Oregon, United States, 97201 Collapse << |
NCT00274248 | Acute Myelogenous Leukemia | Phase 1 | Completed | - | United States, Massachusetts ... more >> The Dana Farber Cancer Institute Boston, Massachusetts, United States, 02134 Collapse << |
NCT00297921 | Acute Myelogenous Leukemia | Phase 1 Phase 2 | Withdrawn | - | - |
实验方案
技术信息
CAS号 | 387867-13-2 | 储存条件 |
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分子式 | C31H42N6O4 | 运输 | 蓝冰 | |||||||||
分子量 | 562.70 | 别名 | MLN518;CT53518;NSC-726292;CT53518 hydrochloride;MLN 518 hydrochloride;坦度替尼 | |||||||||
溶解度 |
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动物实验配方 |
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NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
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NCT00064584 | Acute Myelogenous Leukemia ... more >> Myelodysplastic Syndrome Collapse << | Phase 1 | Completed | - | United States, California ... more >> UCLA Medical Center Los Angeles, California, United States, 90095 United States, Massachusetts Dana Farber Cancer Institute Boston, Massachusetts, United States, 02115 United States, New York Memorial Sloan Kettering Cancer Center New York, New York, United States, 10021 United States, Ohio Ohio State University Medical Center Columbus, Ohio, United States, 43210 United States, Oregon Oregon Health Sciences University Portland, Oregon, United States, 97201 Collapse << |
NCT00274248 | Acute Myelogenous Leukemia | Phase 1 | Completed | - | United States, Massachusetts ... more >> The Dana Farber Cancer Institute Boston, Massachusetts, United States, 02134 Collapse << |
NCT00297921 | Acute Myelogenous Leukemia | Phase 1 Phase 2 | Withdrawn | - | - |
NCT00379080 | Adult Brain Tumor ... more >> Adult Giant Cell Glioblastoma Adult Glioblastoma Adult Gliosarcoma Recurrent Adult Brain Tumor Collapse << | Phase 1 Phase 2 | Completed | - | United States, Alabama ... more >> University of Alabama at Birmingham Birmingham, Alabama, United States, 35294 United States, Florida H. Lee Moffitt Cancer Center and Research Institute Tampa, Florida, United States, 33612 United States, Georgia Emory University Atlanta, Georgia, United States, 30322 United States, Maryland Johns Hopkins University Baltimore, Maryland, United States, 21287 United States, Massachusetts Massachusetts General Hospital Cancer Center Boston, Massachusetts, United States, 02114 Dana-Farber Cancer Institute Boston, Massachusetts, United States, 02115 United States, Michigan Henry Ford Hospital Detroit, Michigan, United States, 48202 United States, North Carolina Wake Forest University Health Sciences Winston-Salem, North Carolina, United States, 27157 United States, Ohio Cleveland Clinic Foundation Cleveland, Ohio, United States, 44195 Collapse << |
NCT00408902 | - | - | Completed | - | - |
NCT00667394 | Glioblastoma ... more >>Gliosarcoma Anaplastic Astrocytoma Anaplastic Oligodendroglioma Anaplastic Mixed Oligoastrocytoma Collapse << | Phase 2 | Completed | - | United States, Maryland ... more >> National Institutes of Health Clinical Center, 9000 Rockville Pike Bethesda, Maryland, United States, 20892 Collapse << |
NCT00390468 | - | - | Completed | - | - |
NCT00390468 | Metastatic Cancer ... more >> Pain Prostate Cancer Collapse << | Phase 2 | Completed | - | United States, Texas ... more >> M. D. Anderson Cancer Center at University of Texas Houston, Texas, United States, 77030-4009 Collapse << |
NCT00379080 | - | - | Completed | - | - |
NCT00408902 | Clear Cell Renal Cell Carcinom... more >>a Recurrent Renal Cell Cancer Stage IV Renal Cell Cancer Collapse << | Phase 2 | Completed | - | United States, Ohio ... more >> Case Western Reserve University Cleveland, Ohio, United States, 44106 Collapse << |
NCT00667394 | - | - | Completed | - | - |
NCT00904852 | Glioblastoma Multiforme | Phase 1 | Withdrawn | June 2010 | - |
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