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CAS No.: 740816-86-8
Synonyms: CGP62221;O-Desmethyl PKC412
O-Desmethyl Midostaurin (CGP62221; O-Desmethyl PKC412) is the active metabolite of Midostaurin (HY-10230) via cytochrome P450 liver enzyme metabolism. O-Desmethyl Midostaurin can be used as an indicator for Midostaurin metabolism in vivo[1]. Midostaurin is a multi-targeted protein kinase inhibitor with IC50 ranging from 22-500 nM.
生物活性
实验方案
技术信息
CAS号 | 740816-86-8 | 储存条件 |
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分子式 | C34H28N4O4 | 运输 | 蓝冰 | |
分子量 | 556.61 | 别名 | CGP62221;O-Desmethyl PKC412 |
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