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CAS No.: 1228013-30-6
Synonyms: CC-223;ATG-008
CC-223 is a potent mTOR kinase inhibitor (IC50=16 nM), with > 150-fold sensitivity over the related lipid kinase PI3Kα (IC50=4 μM).
规格 | 价格 | 促销价格 | 库存 | 数量 |
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生物活性
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
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NCT03591965 | Hepatocellular Carcinoma | Phase 2 | Recruiting | July 1, 2021 | China, Heilongjiang ... more >> Oncology Hospital of Haerbin Medical University Not yet recruiting Harbin, Heilongjiang, China, 150000 Contact: Yuxian Bai bai_yuxian@126.com China, Jiangsu China People PLA 81 Hospital Not yet recruiting Nanjing, Jiangsu, China, 210000 Contact: Shukui Qin 86-25-80864748 qinsk@csco.org.cn China The first Hospital of Jilin University Not yet recruiting Changchun, China Contact: Wei Li jdyylw@163.com Hunan Province Oncology Hospital Not yet recruiting Changsha, China Contact: Sahnzhi Gu 105575191@qq.com Daping Hospital Not yet recruiting Chongqing, China Contact: Dong Wang Dongwang64@hotmail.com The first hospital of Chongqing medical university Not yet recruiting Chongqing, China Contact: Chengyou Du duchengyou@126.com Xiehe Hospital of Fujian Medical University Not yet recruiting Fuzhou, China Contact: Xiaoyan Lin 13950482366@qq.com Nanfang Hospital of Nanfang Medical University Not yet recruiting Guangzhou, China Contact: Yabing Guo gyabing@126.com The first affiliated Hospital of Zhejiang University Not yet recruiting Hangzhou, China Contact: Weijia Fang weijiafang@163.com Zhejiang Province Oncology Hospital Not yet recruiting Hangzhou, China Contact: Jieer Ying jieerying@aliyun.com The first affiliated hospital of Anhui medical university Not yet recruiting Hefei, China Contact: Kangsheng Gu 13805692145@163.com The second affiliated hospital of Anhui medical university Not yet recruiting Hefei, China Contact: Zhengdong Chen chenzhendong@csco.org.cn The first affiliated hospital of Guangxi Medical University Not yet recruiting Nanning, China Contact: Xiaohua Hu gxykdhxh@sina.com Oncology Hospital of Fudan University Not yet recruiting Shanghai, China Contact: Zhiqiang Meng mengfudan2018@yeah.net Zhongshan Hospital of Fudan University Not yet recruiting Shanghai, China Contact: Zhenggang Ren ren.zhenggeng@zs-hospital.sh.cn China PLA general hospital of Shenyang Not yet recruiting Shenyang, China Contact: Zhengdong Zheng Contact mylonzzdong@163.com Tangdu Hospital of China PLA fourth medical university Not yet recruiting Xi'an, China Contact: Helong Zhang zhanghelong@medmail.com.cn Korea, Republic of Dong-A University Hospital Not yet recruiting Busan, Korea, Republic of Contact: Nan-ji Ha 82 51 240 2588 Pusan National Univ. Hospital Not yet recruiting Busan, Korea, Republic of Contact: Jung hee Bark 82 51 240 7079 Kyungpook National Univ. Hospital Not yet recruiting Daegu, Korea, Republic of Contact: Hye-ran Kim 82 53 200 6357 Severance Hospital Recruiting Seoul, Korea, Republic of, 03722 Contact: Kwang-Hyub Han Asan Medical Center Not yet recruiting Seoul, Korea, Republic of Contact: Hye-min Lee 82 2 3010 6280 Seoul National University Hospital Recruiting Seoul, Korea, Republic of Contact: Min-kyoung Kim 82 2 2072 7450 Severance Hospital, Yonsei University Health System Not yet recruiting Seoul, Korea, Republic of Contact: Jung-hee Park Taiwan China Medical University Hospital Recruiting Taichung, Taiwan Contact: Chang-Fang Chiu 04-22053366 ext 5022 d5686@mail.cmuh.org.tw National Taiwan University Hospital Not yet recruiting Taipei, Taiwan Contact: Pei-Jer Chen 02-2312-3456 ext 67072 peijerchen@ntu.edu.tw Taipei Medical University Hospital Recruiting Taipei, Taiwan Contact: Wei-Yu Kao 02-2737 2181 ext 3577 121021@tmuh.org.tw Taipei Veterans General Hospital Recruiting Taipei, Taiwan Contact: Yee Chao 02-28757618 ychao@vghtpe.gov.tw Chang Gung Memorial Hospital-Linkuo Recruiting Taoyuan, Taiwan Contact: Tsai-Sheng Yang 03-328-1200 ext 8825 a481124@adm.cgmh.org.tw Collapse << |
NCT01545947 | Carcinoma, Non-Small-Cell Lung... more >> Non-Small Cell Lung Cancer Collapse << | Phase 1 | Completed | - | United States, California ... more >> Cedars Sinai Medical Center, Inflammatory Bowel Disease Center Los Angeles, California, United States, 90048 University of California, San Francisco San Francisco, California, United States, 9411 United States, New York NYU School of Medicine New York, New York, United States, 10016 United States, South Carolina Cancer Center of the Carolinas Greenville, South Carolina, United States, 29605 United States, Tennessee Henry-Joyce Cancer Clinic Nashville, Tennessee, United States, 37232-5505 United States, Texas Mary Crowley Cancer Research Centers - Medical City Dallas, Texas, United States, 75201 The University of Texas MD Anderson Cancer Center Houston, Texas, United States, 77030 Spain Vall d´Hebron University Hospital Barcelona, Spain, 08035 Hospital Virgen del RocíoServicio de Hematologia Sevilla, Spain, 41013 Collapse << |
NCT02031419 | Lymphoma, Large B-Cell, Diffus... more >>e Collapse << | Phase 1 | Active, not recruiting | November 30, 2020 | United States, California ... more >> Sansum Clinic Santa Barbara, California, United States, 93105 Stanford Cancer Center Stanford, California, United States, 94305 United States, Colorado Rocky Mountain Cancer Centers, LLP [Boulder-COBO] Boulder, Colorado, United States, 80303 United States, Connecticut Yale Cancer Center New Haven, Connecticut, United States, 06510 United States, Florida H. Lee Moffitt Cancer Cencer and Research Institute Tampa, Florida, United States, 33612 United States, Illinois Northwestern University, Division of Hematology Oncology, Dept. of Medicine Chicago, Illinois, United States, 60611 Illinois Cancer Specialists Niles, Illinois, United States, 60714 United States, Minnesota Mayo Clinic Rochester, Minnesota, United States, 55905 United States, Oregon Willamette Valley Cancer Center Eugene, Oregon, United States, 97401-8122 United States, Tennessee West Cancer Center Germantown, Tennessee, United States, 38138 Sarah Cannon Cancer Center Nashville, Tennessee, United States, 37203 United States, Texas MD Anderson Cancer Center Houston, Texas, United States, 77030-400 United States, Wisconsin University of Wisconsin Osteoporosis Clinical Center and Research Program Madison, Wisconsin, United States, 53792 Canada, Alberta Cross Cancer Institute Edmonton, Alberta, Canada, T6G 1Z2 Canada, Ontario Princess Margaret Hospital Toronto, Ontario, Canada, M5G 2M9 France Institut Bergonie Centre Regional de Lutte Contre Le Cancer de Bordeaux Et Sud Ouest Bordeaux, France, 33076 Centre Leon Berard Lyon, France, 69373 Institut Gustave Roussy Villejuif Cedex, France, 94805 Italy Istituto Nazionale Dei Tumori Milano, Italy, 20133 Istituto Clinico Humanitas Rozzano (MI), Italy, 20089 Azienda Sanitaria Ospedaliera San Giovanni Battista Molinette Turin, Italy, 10126 Collapse << |
实验方案
技术信息
CAS号 | 1228013-30-6 | 储存条件 |
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分子式 | C21H27N5O3 | 运输 | 蓝冰 | |||||||
分子量 | 397.47 | 别名 | CC-223;ATG-008 | |||||||
溶解度 |
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动物实验配方 |