CAS No.: 503555-55-3
PHA 408 Catalog No. CSN12718
PHA-408 is a potent, highly selective and ATP-competitive IKB kinase-2 (IKK-2) inhibitor (IC50: 40 nM).
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纯度 & 质量文件
批次:
靶点选择性
生物活性
- 描述
- 参考文献
- [1] Chiang PC, Kishore NN, et al. Combined use of pharmacokinetic modeling and a steady-state delivery approach allows early assessment of IkappaB kinase-2 (IKK-2) target safety and efficacy. J Pharm Sci. 2010 Mar;99(3):1278-87.
- [2] Mbalaviele G, Sommers CD, et al. A novel, highly selective, tight binding IkappaB kinase-2 (IKK-2) inhibitor: a tool to correlate IKK-2 activity to the fate and functions of the components of the nuclear factor-kappaB pathway in arthritis-relevant cells and animal models. J Pharmacol Exp Ther. 2009 Apr;329(1):14-25.
实验方案
- 计算器
- 储存液制备
技术信息
| CAS号 | 503555-55-3 | 储存条件 |
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| 分子式 | C29H27ClFN7O2 | 运输 | 蓝冰 | |
| 分子量 | 560.02 | 别名 |
