CAS No.: 1401223-22-0
PI-1840 Catalog No. CSN15914
Synonyms: PI-1840
PI-1840 is a potent and selective inhibitor for chymotrypsin-like (CT-L) (IC50 value = 27 ± 0.14 nM) over trypsin-like and peptidylglutamyl peptide hydrolyzing (IC50 values > 100 μM) activities of the proteasome.
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纯度 & 质量文件
批次:
靶点选择性
生物活性
- 描述
- 参考文献
- [1] Ozcan S, Kazi A, Marsilio F, et al. Oxadiazole-isopropylamides as potent and noncovalent proteasome inhibitors. J Med Chem. 2013 May 23;56(10):3783-805.
- [2] Kazi A, Ozcan S, et al. Discovery of PI-1840, a novel noncovalent and rapidly reversible proteasome inhibitor with anti-tumor activity. J Biol Chem. 2014 Apr 25;289(17):11906-15.
实验方案
- 计算器
- 储存液制备
技术信息
| CAS号 | 1401223-22-0 | 储存条件 |
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| 分子式 | C22H26N4O3 | 运输 | 蓝冰 | |
| 分子量 | 394.47 | 别名 | PI-1840 |
