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CAS No.: 1062243-51-9

Ro3280 Catalog No. CSN16422

Synonyms: Ro5203280;RO-3280

RO3280 is a potent, highly selective inhibitor of Polo-like kinase 1 (PLK1) with IC50 of 3 nM.

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靶点选择性

生物活性

  • 描述
  • 临床研究
  • NCT号适应症或疾病临床期招募状态预计完成时间地点
    NCT02844816Recurrent Bladder Urothelial C... more >>arcinoma Stage 0a Bladder Urothelial Carcinoma AJCC v6 and v7 Stage 0is Bladder Urothelial Carcinoma AJCC v6 and v7 Stage I Bladder Urothelial Carcinoma AJCC v6 and v7 Collapse <<Phase 2RecruitingFebruary 28, 2020-
    NCT02873195Recurrent Colorectal Carcinoma... more >> Refractory Colorectal Carcinoma Stage IV Colorectal Cancer AJCC v7 Stage IVA Colorectal Cancer AJCC v7 Stage IVB Colorectal Cancer AJCC v7 Collapse <<Phase 2Active, not recruitingNovember 30, 2022United States, Arizona ... more >> Mayo Clinic Hospital Phoenix, Arizona, United States, 85054 Mayo Clinic in Arizona Scottsdale, Arizona, United States, 85259 United States, California City of Hope Comprehensive Cancer Center Duarte, California, United States, 91010 USC / Norris Comprehensive Cancer Center Los Angeles, California, United States, 90033 United States, Georgia Emory University Hospital/Winship Cancer Institute Atlanta, Georgia, United States, 30322 United States, Michigan University of Michigan Comprehensive Cancer Center Ann Arbor, Michigan, United States, 48109 United States, Minnesota Mayo Clinic Rochester, Minnesota, United States, 55905 United States, New York Roswell Park Cancer Institute Buffalo, New York, United States, 14263 United States, North Carolina Duke University Medical Center Durham, North Carolina, United States, 27710 United States, Rhode Island Rhode Island Hospital Providence, Rhode Island, United States, 02903 Collapse <<
    NCT03600701Recurrent Non-Small Cell Lung ... more >>Carcinoma Refractory Lung Non-Small Cell Carcinoma Stage IV Non-Small Cell Lung Cancer AJCC v7 Collapse <<Phase 2RecruitingJuly 17, 2021United States, District of Col... more >>umbia MedStar Georgetown University Hospital Recruiting Washington, District of Columbia, United States, 20007 Contact: Site Public Contact    202-444-2223       Principal Investigator: Stephen V. Liu          United States, Virginia University of Virginia Cancer Center Recruiting Charlottesville, Virginia, United States, 22908 Contact: Site Public Contact    434-243-6303    PAS9E@virginia.edu    Principal Investigator: Richard D. Hall Collapse <<
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实验方案

技术信息

CAS号 1062243-51-9 储存条件
分子式 C27H35F2N7O3 运输 蓝冰
分子量 543.61 别名 Ro5203280;RO-3280

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