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CAS No.: 158876-82-5
Synonyms: UR-12592;Pafinur;Rinialer
Rupatadine is a potent dual PAF/H1 antagonist with Ki of 0.55/0.1 μM (rabbit platelet membranes/guinea pig cerebellum membranes).
生物活性
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|---|---|---|---|---|
NCT03770923 | Rheumatoid Arthritis | Phase 3 | Recruiting | October 2027 | Egypt ... more >> Sherief Abd-Elsalam Recruiting Tanta, Egypt, 35111 Contact: Fedaa Kotkata, Msc Collapse << |
NCT01481909 | Mastocytosis | Phase 2 Phase 3 | Completed | - | Germany ... more >> University Charité Berlin, Germany, 10117 Collapse << |
NCT00162786 | Healthy | Phase 4 | Terminated | - | Netherlands ... more >> Brain and Behaviour Institute Maastricht, Netherlands, 6229 ET Collapse << |
实验方案
技术信息
CAS号 | 158876-82-5 | 储存条件 |
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分子式 | C26H26ClN3 | 运输 | 蓝冰 | |
分子量 | 415.96 | 别名 | UR-12592;Pafinur;Rinialer;Alergoliber;Rupax;卢帕他定 |
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|
NCT03770923 | Rheumatoid Arthritis | Phase 3 | Recruiting | October 2027 | Egypt ... more >> Sherief Abd-Elsalam Recruiting Tanta, Egypt, 35111 Contact: Fedaa Kotkata, Msc Collapse << |
NCT01481909 | Mastocytosis | Phase 2 Phase 3 | Completed | - | Germany ... more >> University Charité Berlin, Germany, 10117 Collapse << |
NCT00162786 | Healthy | Phase 4 | Terminated | - | Netherlands ... more >> Brain and Behaviour Institute Maastricht, Netherlands, 6229 ET Collapse << |
NCT00258141 | Allergy | Phase 4 | Unknown | - | Finland ... more >> Ulappatorin Lääkäriasema Not yet recruiting Espoo, Finland Principal Investigator: Leena Ackermann, MD Koskiklinikka, Tampere Lääkärikeskus Not yet recruiting Tampere, Finland, 33101 Principal Investigator: Ari Karppinen, MD Collapse << |
NCT00199225 | Human Experimentation (Human V... more >>olunteers) Collapse << | Phase 1 | Completed | - | Spain ... more >> Centre de Investigació de Medicaments-Intitut de Recerca-Hospital de la Santa Creu i Sant Pau Barcelona, Spain, 08025 Collapse << |
NCT01605487 | Cold Contact Urticaria | Phase 2 | Completed | - | Germany ... more >> Department of Dermatology and Allergy Charité - Universitätsmedizin Berlin, Charitéplatz 1, Germany, 10117 Berlin Collapse << |
NCT00199251 | Urticaria | Phase 3 | Terminated | - | - |
NCT02358265 | Chronic Urticaria | Phase 3 | Unknown | June 2017 | Germany ... more >> Allergie-Centrum-Charite Recruiting Berlin, Germany, 10117 Contact: Karsten Weller, MD karsten.weller@charite.de Contact: Marcus Maurer, MD marcus.maurer@charite.de Principal Investigator: Karsten Weller, MD Collapse << |
NCT00199238 | Urticaria | Phase 2 | Terminated | - | France ... more >> Hospital Saint Louis Paris Cedex 10, France, 75475 Collapse << |
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