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CAS No.: 1140525-25-2
Synonyms: SB 290157 (trifluoroacetate salt);SB-290157
SB 290157 Trifluoroacetate is the trifluoroacetate form of SB 290157. SB 290157 is a competitive and selective C3aR (anaphylatoxin C3a receptor) antagonist. It blocked C3a-induced C3aR internalization in a concentration-dependent manner and C3a-induced Ca(2+) mobilization in RBL-C3aR cells and human neutrophils with IC(50)s of 27.7 and 28 nM, respectively.
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实验方案
技术信息
CAS号 | 1140525-25-2 | 储存条件 |
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分子式 | C24H29F3N4O6 | 运输 | 蓝冰 | |
分子量 | 526.51 | 别名 | SB 290157 (trifluoroacetate salt);SB-290157 |
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