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CAS No.: 87134-87-0
Synonyms: R-(+)-SCH-23390 maleate;SCH-23390
Potent dopamine receptor antagonist (Ki values are 0.2 nM and 0.3 nM at D1 and D5 receptor sub-types, respectively). Also an agonist at 5-HT1C and 5-HT2C receptors in vitro (Ki values are 6.3 nM and 9.3 nM respectively). Blocks quinpirole-induced Kir3 (GIRK) currents (EC50 = 268 nM) independently of receptors.
生物活性
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|---|---|---|---|---|
NCT02124213 | Healthy | Phase 1 | Completed | - | Sweden ... more >> Karolinska Trial Alliance (KTA) M62 Huddinge, Stockholm, Sweden, SE- 141 86 Collapse << |
实验方案
技术信息
CAS号 | 87134-87-0 | 储存条件 |
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分子式 | C21H22ClNO5 | 运输 | 蓝冰 | |||||
分子量 | 403.86 | 别名 | R-(+)-SCH-23390 maleate;SCH-23390 | |||||
溶解度 |
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动物实验配方 |
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
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NCT02124213 | Healthy | Phase 1 | Completed | - | Sweden ... more >> Karolinska Trial Alliance (KTA) M62 Huddinge, Stockholm, Sweden, SE- 141 86 Collapse << |
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