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CAS No.: 851528-79-5
Synonyms: MBX-8025;RWJ 800025
Seladelpar is selectively exhibits activation of peroxisome proliferator-activated receptor δ (PPARδ) which may has therapeutic activity against dyslipidemia, metabolic syndrome, type 2 diabetes, and non-alcoholic steatohepatitis.
生物活性
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
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NCT02609048 | Primary Biliary Cirrhosis (PBC... more >>) Collapse << | Phase 2 | Terminated(Study stopped early... more >> after review of safety and efficacy demonstrated efficacy proof-of-concept and need for dose reduction.) Collapse << | - | - |
NCT03369002 | Hepatic Impairment | Phase 1 | Completed | - | United States, Colorado ... more >> DaVita Clinical Research Lakewood, Colorado, United States, 80228 United States, Florida Orlando Clinical Research Center Orlando, Florida, United States, 32809 United States, Minnesota DaVita Clinical Research Minneapolis, Minnesota, United States, 55404 United States, Tennessee Vrg & Noccr Knoxville, Tennessee, United States, 37920 Collapse << |
NCT03551522 | NASH - Nonalcoholic Steatohepa... more >>titis Collapse << | Phase 2 | Recruiting | December 31, 2020 | United States, Arizona ... more >> CymaBay Research Site Recruiting Glendale, Arizona, United States, 85306 CymaBay Research Site Recruiting Tucson, Arizona, United States, 85712 United States, California CymaBay Research Site Recruiting Los Angeles, California, United States, 90057 United States, Florida CymaBay Research Site Recruiting Boca Raton, Florida, United States, 33434 CymaBay Research Site Recruiting Lakewood Ranch, Florida, United States, 34211 United States, Mississippi CymaBay Research Site Recruiting Flowood, Mississippi, United States, 39232 United States, Tennessee CymaBay Research Site Recruiting Clarksville, Tennessee, United States, 37040 CymaBay Research Site Recruiting Germantown, Tennessee, United States, 38138 CymaBay Research Site Recruiting Hermitage, Tennessee, United States, 37076 CymaBay Research Site Recruiting Knoxville, Tennessee, United States, 37909 United States, Texas CymaBay Research Site Recruiting Chandler, Texas, United States, 85224 CymaBay Research Site Recruiting Dallas, Texas, United States, 75246 CymaBay Research Site Recruiting Live Oak, Texas, United States, 78233 CymaBay Research Site Recruiting Rollingwood, Texas, United States, 78746 Collapse << |
实验方案
技术信息
CAS号 | 851528-79-5 | 储存条件 |
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分子式 | C21H23F3O5S | 运输 | 蓝冰 | |
分子量 | 444.46 | 别名 | MBX-8025;RWJ 800025 |
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|
NCT02609048 | Primary Biliary Cirrhosis (PBC... more >>) Collapse << | Phase 2 | Terminated(Study stopped early... more >> after review of safety and efficacy demonstrated efficacy proof-of-concept and need for dose reduction.) Collapse << | - | - |
NCT03369002 | Hepatic Impairment | Phase 1 | Completed | - | United States, Colorado ... more >> DaVita Clinical Research Lakewood, Colorado, United States, 80228 United States, Florida Orlando Clinical Research Center Orlando, Florida, United States, 32809 United States, Minnesota DaVita Clinical Research Minneapolis, Minnesota, United States, 55404 United States, Tennessee Vrg & Noccr Knoxville, Tennessee, United States, 37920 Collapse << |
NCT03551522 | NASH - Nonalcoholic Steatohepa... more >>titis Collapse << | Phase 2 | Recruiting | December 31, 2020 | United States, Arizona ... more >> CymaBay Research Site Recruiting Glendale, Arizona, United States, 85306 CymaBay Research Site Recruiting Tucson, Arizona, United States, 85712 United States, California CymaBay Research Site Recruiting Los Angeles, California, United States, 90057 United States, Florida CymaBay Research Site Recruiting Boca Raton, Florida, United States, 33434 CymaBay Research Site Recruiting Lakewood Ranch, Florida, United States, 34211 United States, Mississippi CymaBay Research Site Recruiting Flowood, Mississippi, United States, 39232 United States, Tennessee CymaBay Research Site Recruiting Clarksville, Tennessee, United States, 37040 CymaBay Research Site Recruiting Germantown, Tennessee, United States, 38138 CymaBay Research Site Recruiting Hermitage, Tennessee, United States, 37076 CymaBay Research Site Recruiting Knoxville, Tennessee, United States, 37909 United States, Texas CymaBay Research Site Recruiting Chandler, Texas, United States, 85224 CymaBay Research Site Recruiting Dallas, Texas, United States, 75246 CymaBay Research Site Recruiting Live Oak, Texas, United States, 78233 CymaBay Research Site Recruiting Rollingwood, Texas, United States, 78746 Collapse << |
NCT03602560 | Primary Biliary Cholangitis | Phase 3 | Recruiting | December 2021 | United States, Arizona ... more >> Institute for Liver Health Recruiting Chandler, Arizona, United States, 85224 Contact: Dana Robledo 480-686-8874 drobledo@iliverhealth.org Principal Investigator: Anita Kohli, MD United States, Colorado Univeristy of Colorado Denver and Hospital Recruiting Aurora, Colorado, United States, 80045 Contact: Joselin Gonzalez-Diaz 303-724-1866 joselin.gonzalez-diaz@ucdenver.edu Principal Investigator: Lisa Forman, MD United States, Florida Excel Medical Clinical Trials, LLC Recruiting Boca Raton, Florida, United States, 33434 Contact: Jennifer Olivar 561-756-8206 jolivar@emclinicaltrials.com Principal Investigator: Seth J Baum, MD Florida Reserach Institute Recruiting Lakewood Ranch, Florida, United States, 34211 Contact: Kalina Miller 941-727-7772 kalina.miller@fdhs.com Principal Investigator: Guy W Neff, MD United States, Georgia Digestive Healthcare of Georgia Recruiting Atlanta, Georgia, United States, 30309 Contact: Debeh Legaspi 678-686-5073 dlegaspi@digestivehealthcare.net Principal Investigator: Michael R Galambos, MD United States, Indiana Indianapolis Gastroenterology Research Foundation Recruiting Indianapolis, Indiana, United States, 46237 Contact: Sheila Thompson 317-865-2959 sthompson@indygastro.com Principal Investigator: David C Pound, MD United States, Minnesota Minnesota Gastroenterlogy, P.A. Recruiting Maplewood, Minnesota, United States, 55117 Contact: Gavin Mark 612-870-5597 gavin.mark@mngastro.com Principal Investigator: Donald L Zogg, MD United States, Mississippi Southern Therapy and Advance Research (STAR) LLC Recruiting Jackson, Mississippi, United States, 39216 Contact: Evelyn Arendale 769-251-5674 earendale@jacksonliverandgi.com Principal Investigator: Brian B Borg, MD United States, Missouri Kansas City Research Institute Recruiting Kansas City, Missouri, United States, 64131 Contact: Kelly Vargas 816-759-5274 kvargas@kcresearchinstitute.com Contact: Jeanne Zirkle (816) 759-5274 jzirkle@kcresearchinstitute.com Principal Investigator: Bradley L Freilich, MD United States, New York Concorde Medical Group Recruiting New York, New York, United States, 10016 Contact: Resmi Varughese 212-726-9472 rvarughese@concordemed.com Principal Investigator: Hillel Tobias, MD NYU Langone Health Recruiting New York, New York, United States, 10016 Contact: Kristyn Pierce 646-501-8468 Kristyn.Pierce@nyulangone.org Principal Investigator: Carmen Stanca, MD University of Rochester Medical Center Recruiting Rochester, New York, United States, 14642 Contact: Juliana Posato 585-275-4711 juliana_posato@urmc.rochester.edu Principal Investigator: Jonathan C Huang, DO United States, North Carolina Asheville Gastroenterology Associates, a Division of Digestive Health Partners, P.A. Recruiting Asheville, North Carolina, United States, 28801 Contact: Amber Bartlett 828-254-0881 abartlett@ncdhp.com Principal Investigator: Adam S Zivony, MD United States, Pennsylvania Northeast Clinical Research Center, LLC Recruiting Bethlehem, Pennsylvania, United States, 18017 Contact: Jennifer Jones 610-433-4100 jennifer.jones@necresearch.org Principal Investigator: Adam Peyton, DO United States, Tennessee Gastro One Recruiting Germantown, Tennessee, United States, 38138 Contact: Keosha Henderson 901-682-6540 khenderson@gastro1.com Principal Investigator: Ziad Younes, MD GIA Clinical Trials, LLC Recruiting Knoxville, Tennessee, United States, 37909 Contact: Kathy Karnes 865-558-0687 kkarnes@gihealthcare.com Principal Investigator: Jason Huffman, MD United States, Texas Texas Digestive Disease Consultants Recruiting Fort Worth, Texas, United States, 76104 Contact: Neal Bhakta 817-310-4478 nbhakta@tddctx.com Principal Investigator: Apurva A Modi, MD Baylor College of Medicine Recruiting Houston, Texas, United States, 77030 Contact: Jignesh Patel 713-798-5242 jignesh.patel@bcm.edu Principal Investigator: John M Vierling, MD American Research Corporation at Texas Liver Institute Recruiting San Antonio, Texas, United States, 78215 Contact: MaryLou Hernandez 210-253-3426 mhernandez@txliver.com Principal Investigator: Eric J Lawitz, MD Pinnacle Clinical Research Recruiting San Antonio, Texas, United States, 78229 Contact: Kathy Marotta 210-982-0320 ext 1437 kmarotta@pinnacleresearch.com Principal Investigator: Stephen Harrison, MD United States, Virginia Bon Secours Richmond Community Hospital Recruiting Richmond, Virginia, United States, 23226 Contact: Susan Vollum 804-977-8921 susan_vollum@bshsi.org Principal Investigator: Mitchell L Shiffman, MD Collapse << |
NCT02955602 | Primary Biliary Cirrhosis | Phase 2 | Active, not recruiting | January 2020 | - |
NCT03301506 | Primary Biliary Cirrhosis | Phase 2 Phase 3 | Recruiting | March 2022 | - |
靶点 | Description | IC50 |
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