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CAS No.: 851528-79-5

Seladelpar Catalog No. CSN20554

Synonyms: MBX-8025;RWJ 800025

Seladelpar is selectively exhibits activation of peroxisome proliferator-activated receptor δ (PPARδ) which may has therapeutic activity against dyslipidemia, metabolic syndrome, type 2 diabetes, and non-alcoholic steatohepatitis.

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生物活性

  • 描述
  • 临床研究
  • NCT号适应症或疾病临床期招募状态预计完成时间地点
    NCT02609048Primary Biliary Cirrhosis (PBC... more >>) Collapse <<Phase 2Terminated(Study stopped early... more >> after review of safety and efficacy demonstrated efficacy proof-of-concept and need for dose reduction.) Collapse <<--
    NCT03369002Hepatic ImpairmentPhase 1Completed-United States, Colorado ... more >> DaVita Clinical Research Lakewood, Colorado, United States, 80228 United States, Florida Orlando Clinical Research Center Orlando, Florida, United States, 32809 United States, Minnesota DaVita Clinical Research Minneapolis, Minnesota, United States, 55404 United States, Tennessee Vrg & Noccr Knoxville, Tennessee, United States, 37920 Collapse <<
    NCT03551522NASH - Nonalcoholic Steatohepa... more >>titis Collapse <<Phase 2RecruitingDecember 31, 2020United States, Arizona ... more >> CymaBay Research Site Recruiting Glendale, Arizona, United States, 85306 CymaBay Research Site Recruiting Tucson, Arizona, United States, 85712 United States, California CymaBay Research Site Recruiting Los Angeles, California, United States, 90057 United States, Florida CymaBay Research Site Recruiting Boca Raton, Florida, United States, 33434 CymaBay Research Site Recruiting Lakewood Ranch, Florida, United States, 34211 United States, Mississippi CymaBay Research Site Recruiting Flowood, Mississippi, United States, 39232 United States, Tennessee CymaBay Research Site Recruiting Clarksville, Tennessee, United States, 37040 CymaBay Research Site Recruiting Germantown, Tennessee, United States, 38138 CymaBay Research Site Recruiting Hermitage, Tennessee, United States, 37076 CymaBay Research Site Recruiting Knoxville, Tennessee, United States, 37909 United States, Texas CymaBay Research Site Recruiting Chandler, Texas, United States, 85224 CymaBay Research Site Recruiting Dallas, Texas, United States, 75246 CymaBay Research Site Recruiting Live Oak, Texas, United States, 78233 CymaBay Research Site Recruiting Rollingwood, Texas, United States, 78746 Collapse <<
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技术信息

CAS号 851528-79-5 储存条件
分子式 C21H23F3O5S 运输 蓝冰
分子量 444.46 别名 MBX-8025;RWJ 800025

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