400-920-2911 sales@csnpharm.cn
您的位置 : 首页 / Metabolic Enzyme / P450 / Seviteronel
CAS No.: 1610537-15-9
Synonyms: VT-464;INO-464
VT-464 is a potent CYP17 lyase inhibitor (h-Lyase IC50=69 nM) that demonstrated both exceptional in vitro lyase/hydroxylase selectivity (~10-fold) and oral activity in a hamster model of androgen biosynthesis inhibition.
生物活性
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|---|---|---|---|---|
NCT02445976 | Prostate Cancer | Phase 2 | Active, not recruiting | December 2018 | - |
NCT02130700 | Prostate Cancer | Phase 2 | Completed | - | United States, Maryland ... more >> National Institutes of Health, National Cancer Institute Bethesda, Maryland, United States, 20892 Collapse << |
NCT02012920 | Castration-resistant Prostate ... more >>Cancer CRPC Collapse << | Phase 2 | Active, not recruiting | December 2018 | - |
实验方案
技术信息
CAS号 | 1610537-15-9 | 储存条件 |
|
|
分子式 | C18H17F4N3O3 | 运输 | 蓝冰 | |
分子量 | 399.34 | 别名 | VT-464;INO-464 |
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|
NCT02445976 | Prostate Cancer | Phase 2 | Active, not recruiting | December 2018 | - |
NCT02130700 | Prostate Cancer | Phase 2 | Completed | - | United States, Maryland ... more >> National Institutes of Health, National Cancer Institute Bethesda, Maryland, United States, 20892 Collapse << |
NCT02012920 | Castration-resistant Prostate ... more >>Cancer CRPC Collapse << | Phase 2 | Active, not recruiting | December 2018 | - |
NCT02580448 | Cancer of the Breast ... more >> Breast Cancer Advanced Breast Cancer Metastatic Breast Cancer Male Breast Cancer Triple Negative Breast Cancer ER+ Breast Cancer Collapse << | Phase 1 Phase 2 | Active, not recruiting | May 2019 | - |
NCT02361086 | Castration-resistant Prostate ... more >>Cancer CRPC Collapse << | Phase 1 Phase 2 | Active, not recruiting | June 2018 | United States, Florida ... more >> H. Lee Moffitt Cancer Center and Research Institute Tampa, Florida, United States, 33612 United States, Nebraska Urology Cancer Center Omaha, Nebraska, United States, 68130 United States, North Carolina Duke University Medical Center Durham, North Carolina, United States, 27710 United States, South Carolina Carolina Urologic Research Center Myrtle Beach, South Carolina, United States, 29572 United States, Virginia Virginia Oncology Associates Norfolk, Virginia, United States, 23502 Collapse << |
联系我们
官方电话:400-920-2911
二维码
微信公众号 CSN官网