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CAS No.: 127373-66-4
Synonyms: EI546;LY544349;ONO5046
Sivelestat is a competitive inhibitor of human neutrophil elastase(IC50 = 44 nM and Ki=200 nM) and also inhibits leukocyte elastase obtained from rabbit, rat, hamster and mouse.
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生物活性
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
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NCT00417326 | Community-acquired Pneumonia | Phase 2 | Completed | - | Japan ... more >> Chubu Region Chubu, Japan Chugoku Region Chugoku, Japan Hokkaido Region Hokkaido, Japan Hokuriku Region Hokuriku, Japan Kanto Region Kanto, Japan Kinki Region Kinki, Japan Kyushu Region Kyushu, Japan Shikoku Region Shikoku, Japan Tohoku Region Tohuku, Japan Collapse << |
NCT00219375 | Acute Lung Injury ... more >> Systemic Inflammatory Response Syndrome Collapse << | Phase 4 | Completed | - | Japan ... more >> Chubu Region Facility Chubu, Japan Chugoku Region Facility Chugoku, Japan Hokkaido Region Facility Hokkaido, Japan Hokuriku Regional Facility Hokuriku, Japan Kanto Regional Facility Kanto, Japan Kinki Region Facility Kinki, Japan Kyushu Region Facility Kyushu, Japan Shikoku Region Facility Shikoku, Japan Tohoku Region Facility Tohoku, Japan Collapse << |
NCT01170845 | Esophageal Cancer | Not Applicable | Completed | - | Japan ... more >> Chikara Kunisaki Yokohama, Kanagawa, Japan, 232-0024 Collapse << |
实验方案
技术信息
CAS号 | 127373-66-4 | 储存条件 |
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分子式 | C20H22N2O7S | 运输 | 蓝冰 | |||||||||||
分子量 | 434.46 | 别名 | EI546;LY544349;ONO5046;EI 546 sodium salt hydrate;Elaspol sodium salt hydrate;LY 544349 sodium salt hydrate;西维来司他 | |||||||||||
溶解度 |
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动物实验配方 |
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