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CAS No.: 215543-92-3
SU5402 is potent and selective vascular endothelial growth factor receptor (VEGFR) and fibroblast growth factor receptor (FGFR) inhibitor.
生物活性
实验方案
技术信息
CAS号 | 215543-92-3 | 储存条件 |
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分子式 | C17H16N2O3 | 运输 | 蓝冰 | |
分子量 | 296.32 | 别名 |
Cell Lines | Concentration | Assay Type | Time | Activity Description | Data Sources |
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mouse HER14 cells | - | Function assay | - | Inhibition of EGFR in mouse HER14 cells assessed as inhibition of EGF-stimulated Shc phosphorylation by immunoblotting | 9139660 |
mouse NIH/3T3 cell | - | Function assay | - | Inhibition of acidic FGF-stimulated FGFR1 tyrosine autophosphorylation in mouse NIH/3T3 cells by immunoblottingm, IC50=10 μM | 9139660 |
mouse NIHIR cells | - | Function assay | - | Inhibition of insulin-stimulated insulin receptor beta subunit autophosphorylation in mouse NIHIR cells | 9139660 |
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