CAS No.: 1159101-48-0
Tarafenacin D-tartrate Catalog No. CSN17505
Synonyms: SVT-40776 D-tartrate;Tarafenacin (D-tartrate)
Tarafenacin D-tartrate is a highly selective M3 muscarinic receptor antagonist (Ki= 0.19 nM), ~200 fold selectivity over M2 receptor.
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纯度 & 质量文件
批次:
靶点选择性
生物活性
- 描述
- 参考文献
- [1] Huang X, Zheng G, et al. Microscopic binding of M5 muscarinic acetylcholine receptor with antagonists by homology modeling, molecular docking, and molecular dynamics simulation. J Phys Chem B. 2012 Jan 12;116(1):532-41. doi: 10.1021/jp210579b. Epub 2011 Dec 20.
- [2] Salcedo C, Davalillo S, et al. In vivo and in vitro pharmacological characterization of SVT-40776, a novel M3 muscarinic receptor antagonist, for the treatment of overactive bladder. Br J Pharmacol. 2009 Mar;156(5):807-17.
实验方案
- 计算器
- 储存液制备
技术信息
| CAS号 | 1159101-48-0 | 储存条件 |
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| 分子式 | C25H26F4N2O8 | 运输 | 蓝冰 | |
| 分子量 | 558.48 | 别名 | SVT-40776 D-tartrate;Tarafenacin (D-tartrate) |
