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CAS No.: 903565-83-3
Synonyms: CSG452;R-7201
Tofogliflozin is a potent and highly specific sodium/glucose cotransporter 2 (SGLT2) inhibitor with Ki values of 2.9, 14.9, and 6.4 nM for human, rat, and mouse SGLT2.
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生物活性
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
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NCT02284269 | - | - | Active, not recruiting | - | - |
NCT02528019 | Effects of the DPP-4 Inhibitor... more >>s or SGLT2 Inhibitors on the Protective Actions for Diabetic Complications Collapse << | Phase 4 | Unknown | August 2018 | Japan ... more >> Kurume University Hospital Recruiting Kurume city, Japan, 830-0011 Contact: Nobuhiro Tahara, MD, PhD +81-942-31-7580 ntahara@med.kurume-u.ac.jp Contact: Sho-ichi Yamagishi, MD, PhD +81-942-31-7562 Principal Investigator: Nobuhiro Tahara, MD, PhD Collapse << |
NCT02201004 | Type 2 Diabetes Mellitus | Phase 4 | Completed | - | Japan ... more >> Investigational Site Number 392-028 Adachi-ku, Japan Investigational Site Number 392-007 Atsugi-shi, Japan Investigational Site Number 392-026 Chuoh-ku, Japan Investigational Site Number 392-021 Fukuoka-shi, Japan Investigational Site Number 392-002 Ichihara-shi, Japan Investigational Site Number 392-012 Iruma-shi, Japan Investigational Site Number 392-003 Kawaguchi-shi, Japan Investigational Site Number 392-014 Kitakyusyu-shi, Japan Investigational Site Number 392-027 Kobe-shi, Japan Investigational Site Number 392-004 Koga-shi, Japan Investigational Site Number 392-022 Kunitachi-shi, Japan Investigational Site Number 392-019 Kurume-shi, Japan Investigational Site Number 392-001 Kyoto-shi, Japan Investigational Site Number 392-024 Kyoto-shi, Japan Investigational Site Number 392-006 Matsudo-shi, Japan Investigational Site Number 392-008 Mito-shi, Japan Investigational Site Number 392-030 Musashino-shi, Japan Investigational Site Number 392-029 Okayama-shi, Japan Investigational Site Number 392-017 Otsu-shi, Japan Investigational Site Number 392-011 Sagamihara-shi, Japan Investigational Site Number 392-020 Sakai-shi, Japan Investigational Site Number 392-010 Sapporo-shi, Japan Investigational Site Number 392-016 Sendai-shi, Japan Investigational Site Number 392-018 Shinjuku-ku, Japan Investigational Site Number 392-005 Shizuoka-shi, Japan Investigational Site Number 392-031 Suita-shi, Japan Investigational Site Number 392-015 Sumida-ku, Japan Investigational Site Number 392-023 Sunto-gun, Japan Investigational Site Number 392-013 Tokorozawa-shi, Japan Investigational Site Number 392-025 Yokohama-shi, Japan Collapse << |
实验方案
技术信息
CAS号 | 903565-83-3 | 储存条件 |
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分子式 | C22H26O6 | 运输 | 蓝冰 | |
分子量 | 386.44 | 别名 | CSG452;R-7201 |