CAS No.: 85511-68-8
VU0238441 Catalog No. CSN27595
VU0238441 is a potent agonist of muscarinic acetylcholine receptor M5 with EC50 of 2.1 μM.
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纯度 & 质量文件
批次:
靶点选择性
生物活性
- 描述
- 参考文献
- [1] Bridges TM, Marlo JE, Niswender CM, et al. Discovery of the first highly M5-preferring muscarinic acetylcholine receptor ligand, an M5 positive allosteric modulator derived from a series of 5-trifluoromethoxy N-benzyl isatins. J Med Chem. 2009;52(11):3445-3448.
- [2] Bridges TM, Kennedy JP, Cho HP, et al. Chemical lead optimization of a pan G(q) mAChR M(1), M(3), M(5) positive allosteric modulator (PAM) lead. Part I: Development of the first highly selective M(5) PAM. Bioorg Med Chem Lett. 2010;20(2):558-562.
实验方案
- 计算器
- 储存液制备
技术信息
| CAS号 | 85511-68-8 | 储存条件 |
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| 分子式 | C16H9ClF3NO2 | 运输 | 蓝冰 | |||||||
| 分子量 | 339.70 | 别名 | ||||||||
| 溶解度 |
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动物实验配方 |
