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CAS No.: 122955-13-9
Synonyms: LS190926 dihydrochloride;LS190926 2HCl;XE 991 (hydrochloride)
XE991 2HCl is a potent and selective blocker of KV7 (KCNQ) voltage-gated potassium channels which blocks KV7.2+7.3 (KCNQ2+3) / M-currents (IC50 = 0.6 - 0.98 μM) and KV7.1 (KCNQ1) homomeric channels (IC50 = 0.75 μM) but is less potent against KV7.1/minK channels (IC50 = 11.1 μM).
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CAS号 | 122955-13-9 | 储存条件 |
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分子式 | C26H22Cl2N2O | 运输 | 蓝冰 | |
分子量 | 449.37 | 别名 | LS190926 dihydrochloride;LS190926 2HCl;XE 991 (hydrochloride);XE-991 |
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