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CAS No.: 1169558-38-6
XL413 is a potent and selective Cdc7 inhibitor with an IC50 of 3.7 nM, > 60-fold selectivity against CK2, > 10-fold selectivity against PIM, and > 300-fold selectivity against a panel of over 100 protein kinases.
生物活性
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|---|---|---|---|---|
NCT00838890 | Refractory Hematologic Cancer | Phase 1 Phase 2 | Terminated | - | United States, Florida ... more >> University Of Miami Miami, Florida, United States, 33136 H. Lee Moffitt Cancer Center & Research Institute Tampa, Florida, United States, 33612 United States, Massachusetts Massachusetts General Hospital Boston, Massachusetts, United States, 02114 United States, New York Roswell Park Buffalo, New York, United States, 14263 Collapse << |
NCT00886782 | Advanced Solid Cancers ... more >> Metastatic Cancer Collapse << | Phase 1 Phase 2 | Terminated | - | United States, Massachusetts ... more >> Dana-Farber Cancer Institute Boston, Massachusetts, United States, 02115 United States, Michigan Karmanos Cancer Institute Detroit, Michigan, United States, 48201 Canada, Ontario Local Institution Toronto, Ontario, Canada, M5G 2M9 France Local Institution Villejuif Cedex, France, 94800 Collapse << |
实验方案
技术信息
CAS号 | 1169558-38-6 | 储存条件 |
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分子式 | C14H12ClN3O2 | 运输 | 蓝冰 | |
分子量 | 289.72 | 别名 |
NCT号 | 适应症或疾病 | 临床期 | 招募状态 | 预计完成时间 | 地点 |
---|
NCT00838890 | Refractory Hematologic Cancer | Phase 1 Phase 2 | Terminated | - | United States, Florida ... more >> University Of Miami Miami, Florida, United States, 33136 H. Lee Moffitt Cancer Center & Research Institute Tampa, Florida, United States, 33612 United States, Massachusetts Massachusetts General Hospital Boston, Massachusetts, United States, 02114 United States, New York Roswell Park Buffalo, New York, United States, 14263 Collapse << |
NCT00886782 | Advanced Solid Cancers ... more >> Metastatic Cancer Collapse << | Phase 1 Phase 2 | Terminated | - | United States, Massachusetts ... more >> Dana-Farber Cancer Institute Boston, Massachusetts, United States, 02115 United States, Michigan Karmanos Cancer Institute Detroit, Michigan, United States, 48201 Canada, Ontario Local Institution Toronto, Ontario, Canada, M5G 2M9 France Local Institution Villejuif Cedex, France, 94800 Collapse << |
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