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Adenosine Receptor

Adenosine Receptor

货号 产品名 CAS号 信息
CSN12242 ZM241385 139180-30-6 ZM241385 is a high affinity antagonist ligand selective for the adenosine A2A receptor.
CSN19381 1H-Purine-2,6(3H,7H)-dione 69-89-6 Xanthine is a natural occuring purine-base adenosine receptor antagonist, from which a number of stimulants such as caffeine and theobromine are derived.
CSN18277 Vipadenant 442908-10-3 Vipadenant is an adenosine antagonist with Ki of 1.3 nM and 68 nM for A2A and A1, respectively. Vipadenant is a selective A2A receptor antagonist with Ki values of 1.3, 68, 63, and 1,005 nM for A2A, A1, A2B, and A3 receptors, respectively, used in development for for Parkinson's disease.
CSN13164 Tozadenant 870070-55-6 Tozadenant is a selective adenosine A2A receptor antagonist with Ki values of 11.5 nM on human A2A and 6 nM on rhesus A2A, which can improve motor function in animal models of Parkinson's disease.
CSN11901 SCH58261 160098-96-4 SCH 58261 is a potent and selective A2a adenosine receptor antagonist with Ki of 2.3 nM and 2 nM for rat A2a and bovine A2a, respectively.
CSN15960 Regadenoson 313348-27-5 Regadenoson is a selective adenosine A2A receptor agonist with Ki value of 1.1nM for pig striatum A2A receptor, used as a novel pharmacologic stress agent under clinical development for myocardial perfusion imaging.
CSN11787 Propentofylline 55242-55-2 Propentofylline, a xanthine derivative with purported neuroprotective effects, acts as a c-AMP phosphodiesterase inhibitor, a nerve growth factor stimulator, an adenosine transport inhibitor and a non-selective adenosine receptor antagonist.
CSN12717 Preladenant 377727-87-2 Preladenant is a highly selective and competitive A2A receptor antagonist with Ki value of 1.1nM, used in trials studying the treatment of brain diseases, such as parkinson disease, movement disorders, antipsychotic agents and parkinsonian disorders.
CSN13188 PD 117519 96392-15-3 PD117519 is an adenosine agonist.
CSN16615 Norisoboldine 23599-69-1 Norisoboldine is an isoquinoline alkaloid isolated and purfied from the roots of Lindera aggregata, which acts as an AhR agonist, and enhances the function of the adenosine A1 receptor.
CSN18541 APNEA 89705-21-5 N6-[2-(4-Aminophenyl)ethyl]adenosine is a potent, non-selective A3 adenosine receptor agonist.
CSN11502 N6-Cyclohexyladenosine 36396-99-3 N6-Cyclohexyladenosine is a selective A1 receptor agonist (EC50 = 8.2 nM).
CSN18631 N-[(4-Aminophenyl)methyl]adenosine 95523-13-0 N-[(4-Aminophenyl)methyl]adenosine is an adenosine receptor inhibitor, with Ki of 29 nM for rat ecto-5′-nucleotidase.
CSN18529 LUF6000 890087-21-5 LUF6000 is an allosteric modulator of the human A3 adenosine receptor (AR).
CSN19808 LAS38096 851371-22-7 LAS38096 is a potent, selective, and efficacious A2B adenosine receptor antagonist.
CSN12709 (E)-8-(3,4-Dimethoxystyryl)-1,3-diethyl-7-methyl-3,7-dihydro-1H-purine-2,6-dione 155270-99-8 Istradefylline is a very potent, selective and orally active adenosine A2A receptor antagonist (Ki=2.2 nM) in experimental models of Parkinson's disease.
CSN16958 Piclidenoson 152918-18-8 IB-MECA is an agonist of the adenosine A3 receptor with EC50 values of 0.11 μM. IB-MECA is a potent and selective A3 adenosine receptor agonist with Ki value of 1.1, 54 and 56 nM for A3, A1 and A2A receptors, respectively, which possessing cardioprotective effect and reduces infarct size upon reperfusion in rats.
CSN17618 GR79236 124555-18-6 GR79236 is a highly potent and selective adenosine A1 receptor agonist (Ki = 3.1 nM) that has analgesic and anti-inflammatory actions in humans and animals.
CSN10909 Enprofylline 41078-02-8 Enprofylline is a xanthine derivative used in the treatment of asthma, which acts as a bronchodilator.
CSN10605 3-(4-(2-((6-Amino-9-((2R,3R,4S,5S)-5-(ethylcarbamoyl)-3,4-dihydroxytetrahydrofuran-2-yl)-9H-purin-2-yl)amino)ethyl)phenyl)propanoic acid 120225-54-9 CGS 21680 is an adenosine A2 receptor agonist with IC50 of 22 nM, exhibits 140-fold over A1 receptor.
CSN18682 CGS 21680 HCl 124431-80-7 CGS 21680 HCl is A2A adenosine receptor agonist with Ki value of 27 nM, which can be used to distinguish A2A- and A2B-mediated effect and shows affinity for both A1 and A3 adenosine receptors.
CSN10537 Capadenoson 544417-40-5 Capadenoson is an oral active, potent and selective adenosine A1 receptor agonist.
CSN12871 Theophylline-7-acetic Acid 652-37-9 Acefylline is an adenosine receptor antagonist, a stimulant drug of the xanthine chemical class.
CSN17909 Ab-meca 152918-26-8 AB-MECA is a high affinity A3 adenosine receptor agonist, has high affinity for recombinant A1 and A3 receptors.
CSN17107 (2S,3S,4R,5R)-5-(2-Chloro-6-((3-iodobenzyl)amino)-9H-purin-9-yl)-3,4-dihydroxy-N-methyltetrahydrofuran-2-carboxamide 163042-96-4 2-Cl-IB-MECA is a highly selective A3 adenosine receptor agonist with Ki value of 0.33nM, displaying 2500- and 1400-fold selectivity over A1 and A2A receptors, respectively.
CSN23055 PSB-1115 152529-79-8
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