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GABA Receptor
| 货号 | 产品名 | CAS号 | 信息 |
|---|---|---|---|
| CSN12084 | Tiagabine | 115103-54-3 | Tiagabine is an anti-convulsive medication and a selective gamma-aminobutyric acid (GABA) reuptake inhibitor. |
| CSN12085 | Tiagabine HCl | 145821-59-6 | Tiagabine HCl is an inhibitor of gamma-aminobutyric acid (GABA) reuptake (IC50 = 67 nM in vivo) with anticonvulsant effect. |
| CSN12077 | Thiocolchicoside | 602-41-5 | Thiocolchicoside is a small molecule muscle relaxant and anti-inflammatory agent, shown to function as a competitive GABAA (gamma-aminobutyric acid type A) receptor antagonist. |
| CSN18728 | Propofol | 2078-54-8 | Propofol is a short-acting medication that results in a decreased level of consciousness and lack of memory for events. |
| CSN10515 | Progabide | 62666-20-0 | Progabide is an analog and prodrug of gamma-aminobutyric acid. It is commonly used in the treatment of epilepsy with agonistic activity for both the GABAA and GABAB receptors. Progabide has been investigated for many diseases besides epilepsy, including Parkinson's disease, schizophrenia, clinical depression and anxiety disorder with varying success. |
| CSN11770 | Primidone | 125-33-7 | Primidone is a pyrimidinedione derivative with anticonvulsant activity. |
| CSN11659 | Pazinaclone | 103255-66-9 | Pazinaclone is a sedative and anxiolytic drug in the cyclopyrrolone family of drugs. |
| CSN16621 | NS11394 | 951650-22-9 | NS11394 is a potent and subtype-selective GABA (A) receptor-positive modulator, possessing a functional efficacy selectivity profile of alpha(5) > alpha(3) > alpha(2) > alpha(1) at GABA (A) alpha subunit-containing receptors. |
| CSN11488 | Nefiracetam | 77191-36-7 | Nefiracetam is a neuronal systems enhancer for Ro 5-4864-induced convulsions. Nefiracetam has GABAergic, cholinergic, and monoaminergic properties. |
| CSN10962 | Etifoxine | 21715-46-8 | Etifoxine is potentiator of GABAA receptor function in cultured neurons. |
| CSN13109 | Demoxepam | 963-39-3 | Demoxepam is a drug which is a benzodiazepine derivative. |
| CSN10673 | Clomethiazole | 533-45-9 | Clomethiazole can act as an agonist of GABAA and modulator of glycine receptor. It is a sedative used in the treatment of alcohol withdrawal. |
| CSN11041 | Chlormezanone | 80-77-3 | Chlormezanone can bind to central benzodiazepine receptors, used in the management of anxiety and in the treatment of muscle spasm. |
| CSN10524 | 4-Amino-3-(4-chlorophenyl)butanoic acid | 1134-47-0 | Baclofen, a gamma-amino-butyric acid derivative, is a selective GABAB agonist with IC50 of 200 nM which used as a skeletal muscle relaxant. |
| CSN10266 | Alpidem | 82626-01-5 | Alpidem is a peripheral benzodiazepine GABAA receptor (PBR) ligand and an anxiolytic. |
| CSN10227 | Afloqualone | 56287-74-2 | Afloqualone is an agonist of GABA receptor and has muscle-relaxant effects. |
| CSN10198 | Acamprosate calcium | 77337-73-6 | Acamprosate calcium is an agonist of GABA receptor. It can act as a modulator of glutamatergic systems and reduce alcohol consumption in animal models of alcohol addiction. |
| CSN11821 | (R)-Baclofen HCl | 63701-55-3 | (R)-Baclofen HCl is a derivative of gamma-aminobutyric acid (GABA) primarily used to treat spasticity and is in the early research stages for use for the treatment of alcoholism. |
| CSN10435 | (R)-6-((S)-6-Methyl-5,6,7,8-tetrahydro-[1,3]dioxolo[4,5-g]isoquinolin-5-yl)-[1,3]dioxolo[4,5-e]isobenzofuran-8(6H)-one | 485-49-4 | (+)-Bicuculline is an antagonist of GABAA receptor with IC50 of 2 μM and also shows inhibition of Ca(2+)-activated potassium channels. |
