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HSP
| 货号 | 产品名 | CAS号 | 信息 |
|---|---|---|---|
| CSN16304 | XL888 | 1149705-71-4 | XL888 is a specific and ATP-competitive Hsp90 inhibitor with IC50 of 24 nM. |
| CSN13596 | VER-50589 | 747413-08-7 | VER-50589 is an isoxazole compound that inhibits Hsp90 with an IC50 value of 21 nM. |
| CSN13116 | VER-155008 | 1134156-31-2 | VER-155008 is a potent Hsp70 family inhibitor with IC50 of 0.5 μM, 2.6 μM, and 2.6 μM in cell-free assays for HSP70, HSC70, and GRP78, respectively, > 100-fold selectivity over HSP90. |
| CSN12051 | Teprenone | 6809-52-5 | Teprenone is used as an anti-ulcer drug, a cardioprotective agent, a hepatoprotective agent, a nephroprotective agent, a neuroprotective agent and a Hsp70 inducer. |
| CSN16517 | SNX-2112 | 908112-43-6 | SNX-2112 is a potent synthetic heat shock protein 90 (HSP90) inhibitor with an IC50 of 0.92 μM for K562 cells. |
| CSN15760 | 8-((3,5-Dichlorophenyl)thio)-9-(3-(isopropylamino)propyl)-9H-purin-6-amine | 1454619-14-7 | PU-WS13 is a potent, Grp94-specific Hsp90 inhibitor of the purine scaffold class. |
| CSN16046 | 8-((6-Iodobenzo[d][1,3]dioxol-5-yl)thio)-9-(3-(isopropylamino)propyl)-9H-purin-6-amine | 873436-91-0 | PU-H71 is a potent Hsp90 inhibitor with IC50 of 50 nM. |
| CSN16541 | PF-04929113 | 908115-27-5 | PF-04929113 is a potent and selective HSP90 inhibitor with Kd of 41 nM and induces Her-2 degradation with IC50 of 37 nM. |
| CSN15852 | NVP-HSP990 | 934343-74-5 | NVP-HSP990 is a potent and selective HSP90 inhibitor for HSP90α/β with IC50 of 0.6 nM/0.8 nM. |
| CSN17190 | VER-82576 | 847559-80-2 | NVP-BEP800 is a fully synthetic HSP90β inhibitor with IC50 of 58 nM, exhibits> 70-fold selectivity against Hsp90 family members Grp94 and Trap-1. |
| CSN16765 | NMS-E973 | 1253584-84-7 | NMS-E973 is a potent and selective Hsp90 inhibitor with DC50 of < 10 nM for Hsp90 binding, no activiy against a panel of 52 diverse protein kinases. |
| CSN16562 | KW-2478 | 819812-04-9 | KW-2478 is a nonansamycin HSP90 inhibitor with IC50 of 3.8 nM. |
| CSN11085 | Geldanamycin | 30562-34-6 | Geldanamycin is a natural existing HSP90 inhibitor with Kd of 1.2 μM. |
| CSN15732 | Ganetespib | 888216-25-9 | Ganetespib is a unique triazolone-containing Hsp90 inhibitor with an IC50 of 4 nM in OSA 8 cells. |
| CSN12347 | Elesclomol | 488832-69-5 | Elesclomol, an inhibitor of HSP90, is a potent oxidative stress inducer that elicits pro-apoptosis events among tumor cells. |
| CSN13441 | BIIB021 | 848695-25-0 | BIIB021 is an orally available, fully synthetic small-molecule inhibitor of HSP90 with Ki and EC50 of 1.7 nM and 38 nM, respectively. |
| CSN12421 | Luminespib | 747412-49-3 | AUY922 is a highly potent HSP90 inhibitor for HSP90α/β with IC50 of 13 nM /21 nM, weaker potency against the HSP90 family members GRP94 and TRAP-1. |
| CSN16920 | Onalespib | 912999-49-6 | AT13387 is a selective potent Hsp90 inhibitor with IC50 of 18 nM in A375 cells, displays a long duration of anti-tumor activity. |
| CSN16172 | Alvespimycin | 467214-20-6 | Alvespimycin is a potent, water-soluble HSP90 inhibitor with IC50 of 62 nM. |
