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| 货号 | 产品名 | CAS号 | 信息 |
|---|---|---|---|
| CSN11508 | 6-Carbamimidoylnaphthalen-2-yl 4-guanidinobenzoate dimethanesulfonate | 82956-11-4 | Nafamostat mesylate is a synthetic inhibitor of serine protease with anticoagulant activity. |
| CSN11549 | Milrinone | 78415-72-2 | Milrinone is a phosphodiesterase 3 (PDE3) inhibitor with IC50 of 56 nM, it increases intracellular cyclic adenosine monophosphate resulting in improved ventricular function and vasodilation. |
| CSN11723 | Pimobendan | 74150-27-9 | Pimobendan is a selective inhibitor of PDE3 with IC50 of 0.32 μM. |
| CSN11782 | (8S,9S,10R,13S,14S,17S)-17-Acetyl-10,13-dimethyl-6,7,8,9,10,11,12,13,14,15,16,17-dodecahydro-1H-cyclopenta[a]phenanthren-3(2H)-one | 57-83-0 | Progesterone is an agonist of the nuclear progesterone receptor (nPR)(Kd = 1 nM) and an antagonist of the σ1 receptor. It is involved in many physiological processes such as embryogenesis. |
| CSN11785 | Propafenone HCl | 34183-22-7 | Propafenone HCl, a class I antiarrhythmic drug, is an inhibitor of voltage-dependent sodium channels and treats illnesses associated with rapid heart beats. |
| CSN12096 | Tirofiban | 144494-65-5 | Tirofiban is a non-peptide reversible antagonist of the platelet integrin glycoprotein (GP) IIb/IIIa receptor used as an antiplatelet drug. |
| CSN12189 | 2-(2-Ethoxy-5-((4-ethylpiperazin-1-yl)sulfonyl)phenyl)-5-methyl-7-propylimidazo[5,1-f][1,2,4]triazin-4(1H)-one hydrochloride trihydrate | 330808-88-3 | Vardenafil HCl is a type PDE inhibitor with IC50 of 0.7 and 180 nM for PDE5 and PDE1, respectively. |
| CSN12217 | 2-((4-Chloro-6-((2,3-dimethylphenyl)amino)pyrimidin-2-yl)thio)acetic acid | 50892-23-4 | Wy-14643 is an agonist of PPARα with EC50 of 0.63 μM that can decrease the inflammatory response. It has other functions including lipid metabolism, cell proliferation, differentiation, adipogenesis etc.. |
| CSN12225 | Xylometazoline HCl | 1218-35-5 | Xylometazoline HCl a direct acting sympathomimetic adrenergic α-agonist, used to improve symptoms of nasal congestion, allergic rhinitis, and sinusitis with elimination half-life of >10 seconds. |
| CSN12263 | (S)-5-Chloro-N-((2-oxo-3-(4-(3-oxomorpholino)phenyl)oxazolidin-5-yl)methyl)thiophene-2-carboxamide | 366789-02-8 | Rivaroxaban is an inhibitor of factor Xa (FXa) with IC50 of 0.7 nM and Ki of 0.4 nM which developed for the treatment of thrombotic disease. |
| CSN12278 | Dabigatran | 211914-51-1 | Dabigatran is a reversible and selective, direct thrombin inhibitor (DTI) with Ki value of 4.5 nM. |
| CSN12296 | (Z)-3'-(2-(1-(3,4-Dimethylphenyl)-3-methyl-5-oxo-1H-pyrazol-4(5H)-ylidene)hydrazinyl)-2'-hydroxy-[1,1'-biphenyl]-3-carboxylic acid | 496775-61-2 | Eltrombopag is an agonist of thrombopoietin-receptor (TpoR) and can stimulate thrombopoiesis. |
| CSN12298 | Pravastatin Sodium | 81131-70-6 | Pravastatin Sodium is a competitive HMG-CoA reductase inhibitor with IC50 value of 5.6 μM. |
| CSN12320 | 1-(4-Methoxyphenyl)-7-oxo-6-(4-(2-oxopiperidin-1-yl)phenyl)-4,5,6,7-tetrahydro-1H-pyrazolo[3,4-c]pyridine-3-carboxamide | 503612-47-3 | Apixaban is a direct factor Xa inhibitor with an IC50 of 0.08 nM and 0.17 nM in human and rabbit, respectively. |
| CSN11924 | Sildenafil Citrate | 171599-83-0 | Sildenafil citrate, one of the selective phosphodiesterase-5 (PDE5) inhibitors (IC50= 5.22 nM), is considered the best treatment for erectile dysfunction. |
| CSN11923 | 5-(2-Ethoxy-5-((4-methylpiperazin-1-yl)sulfonyl)phenyl)-1-methyl-3-propyl-1H-pyrazolo[4,3-d]pyrimidin-7(6H)-one | 139755-83-2 | Sildenafil, one of the selective phosphodiesterase-5 (PDE5) inhibitors (IC50= 5.22 nM), is considered the best treatment for erectile dysfunction. |
| CSN11597 | Octreotide acetate | 79517-01-4 | Octreotide acetate is a long-acting octapeptide with pharmacologic actions mimicking those of the natural hormone somatostatin. |
| CSN11512 | Naftopidil | 57149-07-2 | Naftopidil is a selective α1-adrenergic receptor antagonist or α blocker used for treatment for lower urinary tract symptoms (LUTS) due to benign prostatic hyperplasia (BPH). |
| CSN11521 | Naphazoline HCl | 550-99-2 | Naphazoline HCl is a direct-acting sympathomimetic amine with vasoconstrictive activity. |
| CSN12286 | 2-Methyl-6-oxo-1,6-dihydro-[3,4'-bipyridine]-5-carbonitrile 2-hydroxypropanoate(1:x) | 100286-97-3 | Milrinone lactate is a phosphodiesterase 3 (PDE3) inhibitor and a medication used in patients who have heart failure. |
| CSN11969 | (S)-7-((S)-2-(((S)-1-Ethoxy-1-oxo-4-phenylbutan-2-yl)amino)propanoyl)-1,4-dithia-7-azaspiro[4.4]nonane-8-carboxylic acid | 83647-97-6 | Spirapril is an ACE inhibitor antihypertensive drug used to treat hypertension. |
| CSN12097 | (S)-2-(Butylsulfonamido)-3-(4-(4-(piperidin-4-yl)butoxy)phenyl)propanoic acid hydrochloride hydrate | 150915-40-5 | Tirofiban HCl H2O is a non-peptide reversible antagonist of the platelet integrin glycoprotein (GP) IIb/IIIa receptor used as an antiplatelet drug. |
| CSN11719 | Pilsicainide | 88069-67-4 | Pilsicainide is a sodium channel blocker and an antiarrhythmic agent and a drug to treat cardiac arrhythmias in Japan. |
| CSN11510 | Naftidrofuryl | 31329-57-4 | Naftidrofuryl is a vasodilator used in the management of peripheral and cerebral vascular disorders. |
| CSN11603 | 1-((2'-(1H-Tetrazol-5-yl)-[1,1'-biphenyl]-4-yl)methyl)-4-(2-hydroxypropan-2-yl)-2-propyl-1H-imidazole-5-carboxylic acid | 144689-24-7 | Olmesartan is an antagonist of angiotensin II receptor, working as an antihypertensive agent. |
| CSN12057 | Terlipressin | 14636-12-5 | Terlipressin, an analog of vasopressin, acts as vasoconstrictor via V1 receptors on arteriolar smooth muscle cells and can reduce visceral blood flow. It is used to treat hypotension. |
| CSN12190 | Vardenafil HCl | 224785-91-5 | Vardenafil HCl is a PDE5 inhibitor used for treating erectile dysfunction. |
| CSN11481 | Clofibrate | 637-07-0 | Clofibrate, a fibric acid derivative, is a selective agonist of peroxisome proliferator-activated receptor α (PPARα) with EC50 of 50 µM. Clofibrate has been used to treat hyperlipoproteinemia type III and severe hypertriglyceridemia. |
| CSN12174 | Urapidil | 34661-75-1 | Urapidil is a sympatholytic antihypertensive drug. |
| CSN11669 | Penbutolol sulfate | 38363-32-5 | Penbutolol sulfate is able to bind to both beta-1 adrenergic receptors and beta-2 adrenergic receptors (the two subtypes), thus making it a non-selective β blocker. |
| CSN11838 | Revizinone | 133718-29-3 | Revizinone is a selective phosphodiesterase (PDE) inhibitor with IC50 values on this enzyme to 0.036 mM. |
| CSN11458 | Moexipril HCl | 82586-52-5 | Moexipril HCl is a potent orally active non-sulfhydryl angiotensin converting enzyme (ACE) inhibitor, which is used for the treatment of hypertension and congestive heart failure. |
| CSN11605 | Olprinone HCl | 119615-63-3 | Olprinone HCl is a selective phosphodiesterase 3 (PDE3) inhibitor. |
| CSN11643 | Ozagrel sodium | 130952-46-4 | Ozagrel sodium salt is an antiplatelet agent working as a thromboxane A2 synthesis inhibitor. |
| CSN11560 | 5-Isopropyl 3-methyl 2-cyano-6-methyl-4-(3-nitrophenyl)-1,4-dihydropyridine-3,5-dicarboxylate | 75530-68-6 | Nilvadipine is a potent calcium channel blocker with an IC50 of 0.03 nM. |
| CSN52416 | 5-Isopropyl 3-methyl 2-cyano-6-methyl-4-(3-nitrophenyl)-1,4-dihydropyridine-3,5-dicarboxylate | 75530-68-6 | |
| CSN11479 | MRS 2578 | 711019-86-2 | MRS2578 is a potent and selective P2Y6 nucleotide receptor antagonist with IC50 of 37 nM, exhibits insignificant activity at P2Y1, P2Y2, P2Y4,and P2Y11 receptors. |
| CSN11694 | Phentolamine methanesulfonate salt | 65-28-1 | Phentolamine mesylate is a reversible and nonselective alpha-adrenergic receptor antagonist, used for the prevention or control of hypertensive episodes. |
| CSN11784 | Pronethalol | 54-80-8 | Pronethalol is a non-selective beta-adrenergic blocking agent, protect against and to reverse Digitalis-induced ventricular arrhythmias. |
| CSN12117 | Torcetrapib | 262352-17-0 | Torcetrapib is a CETP inhibitor with IC50 of 37 nM, elevates HDL-C and reduces nonHDL-C in plasma. |
| CSN12204 | Vinpocetine | 42971-09-5 | Vinpocetine is a selective inhibitor for PDE1 with IC50 of 21 μM, it also blocks voltage-gated Na+ channels. It's a natural product isolated and purified from the herbs of Catharanthus roseus (L.) G. Don. |
| CSN12233 | 3-(3-((3,4-Dimethoxyphenethyl)(methyl)amino)propyl)-7,8-dimethoxy-4,5-dihydro-1H-benzo[d]azepin-2(3H)-one | 85175-67-3 | Zatebradine is a potent HCN channels antagonist, which decreased the heartbeat in a reversible manner, with 92% inhibition of the hHCN1-mediated current at 10 uM. |
| CSN12305 | (R)-N-(1-(Naphthalen-1-yl)ethyl)-3-(3-(trifluoromethyl)phenyl)propan-1-amine | 226256-56-0 | Cinacalcet is an orally active, second-generation calcimimetic compound and represents a class of compounds for the treatment of hyperparathyroidism. |
| CSN12325 | Prasugrel HCl | 389574-19-0 | Prasugrel HCl is a platelet inhibitor with IC50 value of 1.8 μM. |
| CSN11662 | PD 123319 | 130663-39-7 | PD 123319 is a potent, selective AT2 angiotensin II receptor antagonist with IC50 of 34 nM. |
