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Neurological Disease

货号 产品名 CAS号 信息
CSN11366 1-((4-Chlorophenyl)(phenyl)methyl)-4-(3-methylbenzyl)piperazine dihydrochloride 1104-22-9 Meclizine 2HCl is a histamine H1 receptor antagonist with Ki of 250 nM and is used to treat nausea and motion sickness.
CSN11368 Medetomidine 86347-14-0 Medetomidine is an agonist of α2-adrenoceptor with Ki value of 1.08 nM, used as both a surgical anesthetic and analgesic.
CSN11446 Milnacipran HCl 101152-94-7 Milnacipran HCl is an inhibitor of serotonin-norepinephrine reuptake that can be used to treat fibromyalgia.
CSN11473 Mosapride Citrate 112885-42-4 Mosapride Citrate is both a selective 5HT4 agonist and a 5HT3 antagonist, use as a gastroprokinetic agent.
CSN11489 1-(2-Methylbenzo[d]oxazol-6-yl)-3-(1,5-naphthyridin-4-yl)urea 792173-99-0 SB-334867 free base is a selective non-peptide orexin OX1 receptor antagonist with pKb of 7.2.
CSN11493 (E)-1,2,4-Trimethoxy-5-(prop-1-en-1-yl)benzene 2883-98-9 alpha-Asarone is a naturally occuring inhibitor of both HMG-CoA reductase (IC50 = 3 mM) and certain isoforms of the cytochrome P450 superfamily of enzymes (IC50 = 55.2 and 65.2 μg/ml for CYP2D6 and CYP3A4, respectively), with neuroprotective, anti-oxidative, anticonvulsive and cognitive enhancing action.
CSN11533 Nefopam HCl 23327-57-3 Nefopam HCl, a non-opioid analgesic drug, is blocker of voltage-gated sodium channel and inhibitor of serotonin, dopamine and noradrenaline reuptake. It is used to relieve pain.
CSN11567 Pargyline 555-57-7 Pargyline is an irreversible non-selective monoamine oxidase (MAO) inhibitor drug (IC50 for MAO-A is 11.52 nM and for MAO-B is 8.2 nM) .
CSN11635 4-(Diethylamino)but-2-yn-1-yl 2-cyclohexyl-2-hydroxy-2-phenylacetate 5633-20-5 Oxybutynin a synthetic anticholinergic agent used for treatment of urinary incontinence and overactive bladder syndrome, with elimination half-life of ‎12.4–13.2 hours.
CSN11637 Necrostatin-1 4311-88-0 Necrostatin-1 is an inhibitor of RIP1 and can decrease TNF-α-induced necroptosis with EC50 of 490 nM.
CSN11654 Pargyline HCl 306-07-0 Pargyline HCl is an irreversible and selective MAO-B inhibitor with Ki values of 15 and 1.8 μM for MAO-A and MAO-B, respectively.
CSN11685 Perphenazine 58-39-9 Perphenazine is an inhibitor of 5-HT2A receptor(5-HT2A), alpha-1A adrenergic receptor (α1A), dopamine D2 receptor/dopamine D3 receptor, D2L receptor, and Histamine H1 receptor ( Kis = 5.6, 10, 0.765/0.13, 3.4, and 8 nM respectively). It is commonly used as a typical antipsychotic drug.
CSN11401 Nicardipine HCl 54527-84-3 Nicardipine HCl is a calcium channel blocker that has been widely used to control blood pressure in severe hypertension following events such as ischemic stroke, traumatic brain injury, and intracerebral hemorrhage.
CSN11693 Phenothiazine 92-84-2 Phenothiazine, a dopamine2 (D2) receptor antagonist, could reduce the expression of dopamine in the brain.
CSN11379 Mephenesin 59-47-2 Mephenesin is a centrally acting muscle relaxant which may work as an NMDA receptor antagonist.
CSN11619 Orphenadrine HCl 341-69-5 Orphenadrine HCl is an uncompetitive N-methyl-D-aspartate (NMDA) receptor antagonist with Ki of 6.0 ±0.7 μM.
CSN11657 (3S,4R)-3-((Benzo[d][1,3]dioxol-5-yloxy)methyl)-4-(4-fluorophenyl)piperidine hydrochloride hemihydrate 110429-35-1 Paroxetine HCl is an antidepressant agents known as selective serotonin-reuptake inhibitors (SSRIs).
CSN11451 Mirtazapine 85650-52-8 Mirtazapine is a potent tetracyclic antidepressant.
CSN11360 3-(9,10-Ethanoanthracen-9(10H)-yl)-N-methylpropan-1-amine hydrochloride 10347-81-6 Maprotiline HCl is a bridged-ring tetracyclic antidepressant with adrenergic activity and sedative properties, exerting its effect by blocking the re-uptake of norepinephrine, thereby increasing the synaptic concentration of norepinephrine in the central nervous system and subsequently prolonging the action of norepinephrine on central receptors.
CSN11618 Orphenadrine citrate 4682-36-4 Orphenadrine Citrate is both an uncompetitive NMDA receptor antagonist IC50 value of 16.2 µM and a mAChR antagonist with IC50 value of 0.37 µM.
CSN11417 10-(3-(4-Methylpiperazin-1-yl)propyl)-2-(trifluoromethyl)-10H-phenothiazine dihydrochloride 440-17-5 Trifluoperazine 2HCl is a dopamine D2 receptor inhibitor with anti-dopaminergic and anti-adrenergic actions, which belongs to the phenothiazine compounds.
CSN11477 MPEP 96206-92-7 MPEP is a potent and highly selective non-competitive antagonist at the mGlu5 receptor subtype (IC50 = 36 nM) and a positive allosteric modulator at mGlu4 receptors.
CSN11381 3-(3-Ethyl-1-methylazepan-3-yl)phenol hydrochloride 59263-76-2 Meptazinol HCl is both a partial agonist of μ1 opioid receptor and an AChE inhibitor.
CSN11570 Nomifensine 24526-64-5 Nomifensine is a norepinephrine-dopamine reuptake inhibitor, increases the amount of synaptic norepinephrine and dopamine available to receptors by blocking the dopamine and norepinephrine reuptake transporters.
CSN11659 Pazinaclone 103255-66-9 Pazinaclone is a sedative and anxiolytic drug in the cyclopyrrolone family of drugs.
CSN11501 Memantine 19982-08-2 Memantine is the first in a class of Alzheimer's disease medications acting on the glutamatergic system by blocking NMDA receptors.
CSN11488 Nefiracetam 77191-36-7 Nefiracetam is a neuronal systems enhancer for Ro 5-4864-induced convulsions. Nefiracetam has GABAergic, cholinergic, and monoaminergic properties.
CSN11471 Indeloxazine hydrochloride 65043-22-3 Indeloxazine HCl is an antidepressant and cerebral activator.
CSN11461 Molindone HCl 15622-65-8 Molindone HCl, the salt form of molindone which is a dopamine receptor antagonist, can be used in the treatment of schizophrenia and act as a therapeutic antipsychotic.
CSN11456 Moclobemide 71320-77-9 Moclobemide is a reversible MAO-A inhibitor.
CSN11571 Nomifensine maleate 32795-47-4 Nomifensine maleate is a selective inhibitor of dopamine uptake, used in adult attention deficit disorder.
CSN11688 Phenelzine sulfate 156-51-4 Phenelzine sulfate is a non-selective and irreversible monoamine oxidase inhibitor (MAOI), used as an antidepressant and anxiolytic.
CSN11636 Oxybutynin chloride 1508-65-2 Oxybutynin HCl a synthetic anticholinergic agent used for treatment of urinary incontinence and overactive bladder syndrome, with elimination half-life of ‎12.4–13.2 hours. Oxybutynin HCl is the HCl form of Oxybutynin.
CSN11437 Mianserin 24219-97-4 Mianserin is a H1 receptor inverse agonist and is a psychoactive agent of the tetracyclic antidepressant.
CSN11546 (S)-2-((2S,3S)-2-((S)-2-((S)-1-((2S,3S)-2-((S)-2,6-Diaminohexanamido)-3-methylpentanoyl)pyrrolidine-2-carboxamido)-3-(4-hydroxyphenyl)propanamido)-3-methylpentanamido)-4-methylpentanoic acid 92169-45-4 Neuromedin N is a potent modulator of dopamine D2 receptor agonist binding in rat neostriatal membranes.
CSN11459 Mofegiline HCl 120635-25-8 Mofegiline HCl is a potent and selective enzyme-activated irreversible inhibitor of MAO-B and shows marked selectivity for the B form (IC50 = 680 and 3.6 nM for MAO-A and MAO-B).
CSN11400 Nicardipine 55985-32-5 Nicardipine is a calcium channel blocker that has been widely used to control blood pressure in severe hypertension following events such as ischemic stroke, traumatic brain injury, and intracerebral hemorrhage.
CSN11527 Miglustat 72599-27-0 Miglustat is an inhibitor of glucosylceramide synthase, primarily to treat Type I Gaucher disease (GD1).
CSN11347 LY341495 201943-63-7 LY341495 is a highly potent and selective group II metabotropic glutamate receptor antagonist.
CSN11447 4-Methyl-N-(2-morpholinoethyl)-6-phenylpyridazin-3-amine dihydrochloride 25953-17-7 Minaprine 2HCl is a reversible inhibitor of MAO-A, also weakly inhibits acetylcholinesterase and is an antidepressant for treatment of depression.
CSN11490 1-(2-Methylbenzo[d]oxazol-6-yl)-3-(1,5-naphthyridin-4-yl)urea hydrochloride 249889-64-3 SB-334867 is a selective non-peptide orexin OX1 receptor antagonist with a pKb value of 7.2.
CSN11494 PNU-120596 501925-31-1 PNU-120596 is a a type II positive allosteric modulator of α7 nAChRs with an EC50 of 0.2 μM.
CSN11502 N6-Cyclohexyladenosine 36396-99-3 N6-Cyclohexyladenosine is a selective A1 receptor agonist (EC50 = 8.2 nM).
CSN11528 Miglustat HCl 210110-90-0 Miglustat HCl is an inhibitor of glucosylceramide synthase, primarily to treat Type I Gaucher disease (GD1).
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