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| 货号 | 产品名 | CAS号 | 信息 |
|---|---|---|---|
| CSN10032 | 3-(Hexyloxy)-4-(1-methyl-1,2,5,6-tetrahydropyridin-3-yl)-1,2,5-thiadiazole | 131986-45-3 | Xanomeline is a functionally selective M1/M4 agonist, used in the study of both Alzheimer's disease and schizophrenia. |
| CSN10054 | 5-Chloro-7-iodoquinolin-8-ol | 130-26-7 | Clioquinol is an antifungal drug and antiprotozoal compound that shows effectivity for Alzheimer's disease treatment and induce cancer cell death. |
| CSN10082 | Dibucaine HCl | 61-12-1 | Dibucaine HCl is an anesthetic mainly used for surface anesthesia. |
| CSN10189 | Paliperidone | 144598-75-4 | Paliperidone is a potent serotonin-2A and dopamine-2 receptor antagonist, it is the main active metabolite of risperidone and used in the treatment of schizophrenia. |
| CSN10196 | Piperidin-1-yl(quinoxalin-6-yl)methanone | 154235-83-3 | Ampalex is a positive allosteric modulator of AMPAR and is researched as a treatment for Alzheimer's disease. |
| CSN10208 | 2-Acetoxy-N,N,N-trimethylethanaminium chloride | 60-31-1 | Acetylcholine chloride is a neurotransmitter that can induce the opening of calcium channels. |
| CSN10243 | Alizapride HCl | 59338-87-3 | Alizapride HCl is a dopamine receptor antagonist used in the administration of nausea and vomiting. |
| CSN10289 | Amitriptyline HCl | 549-18-8 | Amitriptyline HCl is a multiple-target molecular as an inhibitor of both 5-HT and NA reuptake (SNRI), and also a TrkA/B agonist. |
| CSN21185 | SR17018 | 2134602-45-0 | SR17018 is brain-penetrant μ-opioid receptor agonist EC50 of 97 nM. |
| CSN21106 | Pimozide | 2062-78-4 | Pimozide is a dopamine receptor antagonist, with Kis of 1.4 nM, 2.5 nM and 588 nM for dopamine D2, D3 and D1 receptors, respectively, and also has affinity at α1-adrenoceptor, with a Ki of 39 nM; also inhibits STAT3 and STAT5. |
| CSN10171 | 7,8-Dihydroxy-2-phenyl-4H-chromen-4-one | 38183-03-8 | 7,8-Dihydroxyflavone acts as an agonist of TrkB receptor with Kd of 320 nM with neuroprotective effect. |
| CSN17907 | Nalfurafine hydrochloride | 152658-17-8 | Nalfurafine HCl is a moderately selective kappa opioid receptor agonist. |
| CSN10227 | Afloqualone | 56287-74-2 | Afloqualone is an agonist of GABA receptor and has muscle-relaxant effects. |
| CSN10072 | N-Benzyl-N,N-dimethyl-2-(2-(4-(2,4,4-trimethylpentan-2-yl)phenoxy)ethoxy)ethanaminium chloride | 121-54-0 | Benzethonium chloride can inhibit nAChRs with IC50 values of 49 nM and 122 nM for α4β2 nAChRs and α7 nAChRs, respectively. It is a synthetic quaternary ammonium salt with surfactant, antiseptic, and broad spectrum antimicrobial properties. |
| CSN10181 | NU1025 | 90417-38-2 | NU1025 is a potent PARP inhibitor with IC50 of 400 nM. |
| CSN10107 | 2-(Diethylamino)ethyl 4-aminobenzoate hydrochloride | 51-05-8 | Procaine HCl is a local anesthetic drug of the amino ester group. |
| CSN10198 | Acamprosate calcium | 77337-73-6 | Acamprosate calcium is an agonist of GABA receptor. It can act as a modulator of glutamatergic systems and reduce alcohol consumption in animal models of alcohol addiction. |
| CSN10249 | Almotriptan malate | 181183-52-8 | Almotriptan Malate a serotonin 5HT-1B/1D-receptor agonist with high affinity for the 5-HT(1B) and 5-HT(1D) receptors, used to treat migraine. |
| CSN10242 | Alizapride | 59338-93-1 | Alizapride is a dopamine antagonist with prokinetic and antiemetic effects used in the treatment of nausea and vomiting, including postoperative nausea and vomiting. |
| CSN10104 | Pizotifen malate | 5189-11-7 | Pizotifen Malate is a benzocycloheptene-based drug used to reduce the frequency of recurrent migraine headacheswith, with high affinity for 5-HT and dopamine receptors (Kis = 7.94 and 2.4 nM for 5-HT2C and D2, respectively). |
| CSN18095 | Olcegepant | 204697-65-4 | Olcegepant is the first potent and selective non-peptide antagonist of the calcitonin gene-related peptide 1 (CGRP1) receptor (IC50= 0.03 nM). |
| CSN10126 | Pizotifen | 15574-96-6 | Pizotifen is a highly selective 5-HT receptor blocking agent, which is a benzocycloheptane based drug. |
| CSN10256 | Eliprodil | 119431-25-3 | Eliprodil can antogonize GluN2B-selective NMDA in a non-competitive manner with IC50 value of 1 μM. It is also a σ1 ligand with Ki value of 0.013 μM. |
| CSN10153 | 5-(2-Aminoethyl)benzene-1,2,4-triol hydrobromide | 636-00-0 | Oxidopamine hydrobromide is a selective catecholaminergic neurotoxin, depletes brain catecholamine levels via uptake and accumulation by a transport mechanism specific to these neurons. |
| CSN10250 | Almotriptan | 154323-57-6 | Almotriptan is a 5-HT1B/1D-receptor agonist used to treat migraine. |
| CSN10132 | Varenicline HCl | 230615-23-3 | Varenicline HCl is a nicotinic receptor partial agonist and it stimulates nicotine receptors more weakly than nicotine itself does. |
| CSN10154 | Oxidopamine HCl | 28094-15-7 | Oxidopamine HCl is a neurotoxic synthetic organic compound, selectively destroys dopaminergic and noradrenergic neurons in the brain. |
| CSN19071 | PF-CBP1 HCl | 2070014-93-4 | PF-CBP1 HCl is a highly selective inhibitor of the bromodomain of CREB-binding protein (CREBBP).It inhibits CREBBP and p300 bromodomains with IC50 of 125 and 363 nM respectively. |
| CSN17659 | (5S,6S,9R)-5-Amino-6-(2,3-difluorophenyl)-6,7,8,9-tetrahydro-5H-cyclohepta[b]pyridin-9-yl 4-(2-oxo-2,3-dihydro-1H-imidazo[4,5-b]pyridin-1-yl)piperidine-1-carboxylate | 1289023-67-1 | BMS-927711 is a highly potent, oral calcitonin gene-related peptide (CGRP) receptor antagonist with a Ki value of 0.027 nM. |
| CSN10099 | Nialamide | 51-12-7 | Nialamide is a non-selective, irreversible monoamine oxidase inhibitor (MAOI) of the hydrazine class that was used as an antidepressant. |
| CSN10182 | NSC-87877 disodium | 56932-43-5 | NSC 87877 is a cell-permeable inhibitor of both SHP-1 and SHP-2 with IC50 values of 355 and 318 nM respectively. It also inhibits EGF-induced Erk1/2 activation in HEK293 cells and significantly reduces MDA-MB-468 cell viability/proliferation. |
